Drug Name Brand Names Drug Class Indications Mechanism of Action
Arformoterol tartrate Brovana Long-Acting beta-2 adrenergic agonist (LABA); Bronchodilator Chronic Obstructive Pulmonary Disease Selective long-acting beta-2 adrenergic receptor agonist, which produces relaxation of bronchial smooth muscle fibers leading to bronchodilation. It is the (R,R)-entantiomer of formoterol, and has a two-fold greater potency of racemic formoterol.
Bitolterol mesylate* * Tornalate (No longer available in the United States) Long-Acting beta-2 adrenergic agonist (LABA); Bronchodilator Asthma; COPD (off-label)  
Formoterol fumarate Foradil Aerolizer; Perforomist Long-Acting beta-2 adrenergic agonist (LABA); Bronchodilator Asthma; Exercise induced asthma prophylaxis; COPD Selective long-acting beta-2 adrenergic agonist which causes an increase in cyclic-AMP by stimulating intracellular adenyl cyclase. This action results in smooth muscle relaxation and inhibition of inflamatory mediators.
Salmeterol xinafoate Serevent Diskus; Serevent HFA Long-Acting beta-2 adrenergic agonist (LABA); Bronchodilator Asthma; Exercise induced asthma prophylaxis; COPD Selectively stimulates the beta-2 adrenergic receptors of intracellular adenyl cyclase, the catalyst for the conversion of adenosine triphosphate (ATP) to cyclic-1’,5’-adenosine monophosphate (cyclic AMP). This action causes an increase in cyclic AMP levels resulting in bronchial smooth muscle relaxation, and inhibition of the release of immediate hypersensitivity mediators from the mast cells.